Des-Arg10-Kallidin

Product Description

Des-Arg10-Kallidin
Catalog number: MDP0673
CAS Number: 183449-57-2
Sequence: Lys-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe . 2AcOH . 4H2O
Amount: 5 mg
Molecular Weight: 1032 g/mol
Supplied as: Powder
Applications: molecular tool for various biochemical applications
Storage: -20 °C
WARNING: For in vitro Research Use Only. NOT for use on humans or animals.
Grade: Biotechnology grade. All products are highly pure.

References:
1: Galizzi JP, Bodinier MC, Chapelain B, Ly SM, Coussy L, Giraud S, Neliat G, Jean T. Up-regulation of [3H]-des-Arg10-kallidin binding to the bradykinin B1 receptor by interleukin-1 beta in isolated smooth muscle cells: correlation with B1 agonist-induced PGI2 production Br J Pharmacol. 1994 Oct;113(2):389-94.
2: Guevara-Lora I, Labedz A, Skrzeczynska-Moncznik J, Kozik A. Bradykinin and des-Arg10-kallidin enhance the adhesion of polymorphonuclear leukocytes to extracellular matrix proteins and endothelial cells Cell Commun Adhes. 2011 Aug;18(4):67-71.
3: Romero JR, Rivera A, Lança V, Bicho MD, Conlin PR, Ricupero DA. Na+/Ca2+ exchanger activity modulates connective tissue growth factor mRNA expression in transforming growth factor beta1- and Des-Arg10-kallidin-stimulated myofibroblasts J Biol Chem. 2005 Apr 15;280(15):14378-84.
4: Schanstra JP, Bataillé E, Marin Castaño ME, Barascud Y, Hirtz C, Pesquero JB, Pecher C, Gauthier F, Girolami JP, Bascands JL. The B1-agonist [des-Arg10]-kallidin activates transcription factor NF-kappaB and induces homologous upregulation of the bradykinin B1-receptor in cultured human lung fibroblasts J Clin Invest. 1998 May 15;101(10):2080-91.
5: Lin KS, Amouroux G, Pan J, Zhang Z, Jenni S, Lau J, Liu Z, Hundal-Jabal N, Colpo N, Bénard F. Comparative studies of three 68Ga-labeled [Des-Arg10]kallidin derivatives for imaging bradykinin B1 receptor expression with PET J Nucl Med. 2015 Apr;56(4):622-7.
6: Amouroux G, Pan J, Jenni S, Zhang C, Zhang Z, Hundal-Jabal N, Colpo N, Liu Z, Bénard F, Lin KS. Imaging Bradykinin B1 Receptor with 68Ga-Labeled [des-Arg10]Kallidin Derivatives: Effect of the Linker on Biodistribution and Tumor Uptake Mol Pharm. 2015 Aug 3;12(8):2879-88.
7: Nowak W, Goldschmidt ED, Falcioni AG, Pugliese MI, Errasti AE, Pelorosso FG, Daray FM, Gago JE, Rothlin RP. Functional evidence of des-Arg10-kallidin enzymatic inactivating pathway in isolated human umbilical vein Naunyn Schmiedebergs Arch Pharmacol. 2007 May;375(3):221-9.
8: Qadri F, Bader M. Kinin B1 receptors as a therapeutic target for inflammation Expert Opin Ther Targets. 2018 Jan;22(1):31-44.
9: Zubakova R, Gille A, Faussner A, Hilgenfeldt U. Ca2+ signalling of kinins in cells expressing rat, mouse and human B1/B2-receptor Int Immunopharmacol. 2008 Feb;8(2):276-81.
10: MacNeil T, Feighner S, Hreniuk DL, Hess JF, Van der Ploeg LH. Partial agonists and full antagonists at the human and murine bradykinin B1 receptors Can J Physiol Pharmacol. 1997 Jun;75(6):735-40.

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